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CRO Business
Assay Developmen
t
High Throughput Screening
Lead Identification
Kinase Assay
GPCR Drug Discovery
Ion Channel Study
Products
cDNA Collection
Cell Lines Collection
Natural Compound Library
Mycoplasma Detection Kit
Wash Free Calcium Assay Kit
Peptide & Peptide Library
Cell Line List
Receptor
Subtype
Description
/
Name
Assay application
Adrenergic
¦Á1AR
HEK293/¦Á1AR
calcium
¦Á2AR
HEK293/¦Á2AR
calcium
¦Á2BR
HEK293/¦Á2BR
calcium
¦Á2CR
HEK293/¦Á2CR
calcium
¦Â2R
CHO or HEK293/CRE/d2EGFP/¦Â2R
EGFP/cAMP
¦Â3R
HEK293/¦Â3R
calcium/cAMP
Calcitonin
CTR
HEK293/CTR/CRE/d2EGFP
EGFP/cAMP
Cholecystokinin
CCKAR
HEK293/CCKAR
calcium
Corticotrophin releasing factor
CRFR1
HEK293/CRFR1
cAMP
CRFR2
HEK293/CRFR2
cAMP
Dopamine
D1R
HEK293/D1R/CRE/¦Â-lactamase
¦Â-lactamase/cAMP
D2R
HEK293/D2R/Ga15
calcium
D5R
HEK293/D5R/CRE/¦Â-lactamase
¦Â-lactamase/cAMP
Galanin
GALR1
HEK293/GALR1
calcium
GALR3
HEK293/GALR3
calcium
Gonadotrophin-releasing hormone
GnRHR
HEK293/GnRHR/NFAT/¦Â-lactamase
¦Â-lactamase/calcium
Free fatty acid
GPR40
HEK293/GPR40/NFAT/¦Â-lactamase
¦Â-lactamase/calcium
GPR120
HEK293/GPR120/NFAT/¦Â-lactamase
¦Â-lactamase/calcium
Histamine
H1R
HEK293/H1R/NFAT/¦Â-lactamase
¦Â-lactamase/calcium
H2R
HEK293/H2R/CRE/¦Â-lactamase
¦Â-lactamase/cAMP
HEK293/H2R/CRE/luciferase
luciferase/cAMP
H3R
HEK293/H3R/Ga15
cAMP/calcium
HEK293/H3R/CRE/luciferase
luciferase/cAMP
H4R
HEK293/H4R/Ga16
cAMP/calcium
5-Hydroxytryptamine
5HT7R
CHO/5HT7R/CRE/bla
¦Â-lactamase/cAMP
Melanocortin
MC4R
HEK293/MC4R/CRE/d2EGFP
EGFP/cAMP
Melanin-concentration hormone
MCHR1
HEK293/MCHR1
calcium/cAMP
MCHR2
HEK293/MCHR2
calcium
Melatonin
MTNR1B
HEK293/MTNR1B
calcium
Muscarinic
M1R
HEK293/M1R
calcium
Neuropeptide
NPYR1
HEK293/NPYR1
calcium
NPYR2
HEK293/NPYR2
calcium
Parathyroid hormone
PTHR1
HEK293/PTHR1/CRE/d2EGFP
EGFP/cAMP
HEK293/PTHR1/CRE/¦Â-lactamase
¦Â-lactamase/cAMP
PTHR2
HEK293/PTHR2/CRE/¦Â-lactamase
¦Â-lactamase/cAMP
Platelet activating factor
PAFR
HEK293/PAFR/NFAT/¦Â-lactamase
¦Â-lactamase/calcium
Substance P
SPR
HEK293/SPR
calcium
For functional assay ion channel cell lines, please contact us for the details.
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