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In House GPCR Collection at HD Biosciences (partial) |
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GPCR Family |
Target |
GPCR Family |
Target |
| Adenosine |
ADORA1 |
Metabotropic Glutamate |
mGluR1 |
| ADORA2A |
mGluR2 |
| ADORA2B |
mGluR3 |
| ADORA3 |
mGluR4 |
| Adrenergic |
Alpha-1A |
mGluR5 |
| Alpha-1B |
mGluR5a |
| Alpha-1D |
mGluR6 |
| Alpha-2A |
mGluR7 |
| Alpha-2B |
mGluR8 |
| Alpha-2B |
Muscarinic |
M1 |
| Beta-2 |
M2 |
| Beta-3 |
M3 |
| Angiotensin |
AT1 |
M5 |
| Bombesin |
BB3 |
Melanin-Concentrating Hormone |
MCH1R |
| Bradykinin |
B1 |
MCH2R |
| B2 |
MAS-related GPR, member D |
MrgD |
| Cannabinoid |
CB2 |
Neuropeptide FF |
NPFF1R |
| Calcitonin |
CTR1 |
Neuropeptide Y |
NPY1R |
| Cholecystokinin |
CCKAR |
NPY2R |
| CCKBR |
Neuromedin U |
NMU1 |
| Corticotropin-Releasing hormone |
CRHR2 |
Opioid |
MU |
| Dopamine |
D1 |
ORL1 |
| D2L |
Orexin |
OX1 |
| D2S |
Platelet-activating factor |
RAF |
| D5 |
Parathyroid Hormone |
PTHR1 |
| Endothelin |
ETB |
PYHR2 |
| Free Fatty Acid |
GPR40 |
Serotonin |
5-HT1A |
| GPR119 |
5-HT2A |
| GPR120 |
5-HT2B |
| Bile acid |
GPR131 |
5-HT2C |
| Galanin |
GALR1 |
Growth hormone secretagoguo |
GHSR1a |
| GALR2 |
Protease-activated receptors |
PAR1 |
| Glucagon |
GCGR |
PAR2 |
| GLP-1 |
PAR4 |
| Gonadotrophin-releasing hormone |
GnRH |
Somatostatin |
sst1 |
| Histamine |
H1 |
sst2 |
| H2 |
sst3 |
| H3 |
sst4 |
| H4 |
sst5 |
| Melatonin |
MT1 |
Tachykinin |
NK1 |
| MT2 |
sNK3 |
| Melanocortin |
MC1R |
Vasopressin |
V1a |
| MC2R |
V1b |
| MC3R |
Urotensin |
UT |
| MC4R |
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